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Home - Products - GPCR/G Protein - Prostaglandin Receptor - AH 6809

AH 6809

CAS No. 33458-93-4

AH 6809( —— )

Catalog No. M24276 CAS No. 33458-93-4

AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    AH 6809
  • Note
    Research use only, not for human use.
  • Brief Description
    AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively).
  • Description
    AH 6809 is an antagonist of EP and DP receptor(with Kis of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively). AH 6809 has a Ki of 350 nM for mouse EP2 receptor.
  • In Vitro
    AH 6809 (1?μM; 30 min) inhibits T. serrulatus venom (TsV)-induced and PGE2-amplified IL-1β and cAMP production in macrophages.AH 6809 (30-300 μM) antagonizes the anti-aggregatory activity of PGD2 in whole blood, with an apparent pA2 of 5.35.
  • In Vivo
    AH 6809 (5 mg/kg; i.p.) decreases TsV-induced mortality, PGE2 and IL-1β production and neutrophil infiltration in the lungs of mice.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Prostaglandin Receptor
  • Recptor
    DP|EP1|EP2|EP3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    33458-93-4
  • Formula Weight
    298.29
  • Molecular Formula
    C17H14O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:25 mg/mL (83.81 mM; Need ultrasonic);H2O:< 0.1 mg/mL (insoluble)
  • SMILES
    CC(C)Oc(cc1)cc(Oc(cc2)c3cc2C(O)=O)c1C3=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

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